PQR620
Ligand Summary
Name: PQR620
PubChem: 121334520
Guide to Pharmacology: 10142
ChEMBL: CHEMBL4286698
LyCHI: 4XWLPHDFK892
Target Activities
MTOR
Serine/threonine-protein kinase mTOR
6 Activities
Items per page:
1 – 6 of 6
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 9.57 | |||||
Ki | 7.97 | |||||
Kd | 9.57 | J Med Chem, (2018) 61:22:10084 | ||||
Kd | 9.57 | J Med Chem, (2019) 62:18:8609 | ||||
Ki | 7.97 | J Med Chem, (2018) 61:22:10084 | ||||
Ki | 7.97 | J Med Chem, (2019) 62:18:8609 | ||||
PIK3CA
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
2 Activities
PIK3C3
Phosphatidylinositol 3-kinase catalytic subunit type 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 5.56 | |||||