CHEMBL566598
Ligand Summary
Name: 7-(6-methoxypyridin-3-yl)-3-(2-oxo-2-(pyrrolidin-1-yl)ethylamino)-1-(2-propoxyethyl)pyrido[3,4-b]pyrazin-2(1H)-one
PubChem: 11993465
ChEMBL: CHEMBL566598
LyCHI: 4DP27R5611F1
Target Activities
PDE5A
cGMP-specific 3',5'-cyclic phosphodiesterase
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 10.1 | Bioorg. Med. Chem. Lett., (2009) 19:17:5209 | ||||
PDE6A
Rod cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.4 | Bioorg. Med. Chem. Lett., (2009) 19:17:5209 | ||||