splitomicin
Ligand Summary
Name: splitomicin
PubChem: 5269
Guide to Pharmacology: 8101
ChEMBL: CHEMBL86537
LyCHI: 4CGURH71RALJ
Target Activities
SIRT1
NAD-dependent protein deacetylase sirtuin-1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 4.02 | |||||
CYP1A2
Cytochrome P450 1A2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
AC50 | 6.3 | None, None:None:None | ||||
CYP2C19
Cytochrome P450 2C19
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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AC50 | 7.1 | None, None:None:None | ||||