NI-57
Ligand Summary
Name: NI-57
PubChem: 91827373
Guide to Pharmacology: 8573
ChEMBL: CHEMBL3752151
LyCHI: 4BTDZRWX2SR3
Target Activities
BRPF1
Peregrin
9 Activities
Items per page:
1 – 9 of 9
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.51 | |||||
IC50 | 8.51 | J Med Chem, (2017) 60:16:6998 | ||||
Kd | 7.51 | MedChemComm, (2015) 6:9:1587 | ||||
Kd | 7.51 | J. Med. Chem., (2016) 59:4:1271 | ||||
Kd | 7.51 | J Med Chem, (2017) 60:16:6998 | ||||
Kd | 7.51 | MedChemComm, (2016) 7:12:2246 | ||||
IC50 | 7.33 | Journal of Medicinal Chemistry, (2017) None:16:6998 | ||||
IC50 | 7.16 | J Med Chem, (2017) 60:16:6998 | ||||
IC50 | 6.94 | J Med Chem, (2017) 60:16:6998 | ||||
BRPF3
Bromodomain and PHD finger-containing protein 3
8 Activities
Items per page:
1 – 8 of 8
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 6.39 | |||||
IC50 | 6.85 | J Med Chem, (2017) 60:16:6998 | ||||
Kd | 6.39 | MedChemComm, (2015) 6:9:1587 | ||||
Kd | 6.39 | J. Med. Chem., (2016) 59:4:1271 | ||||
Kd | 6.39 | J Med Chem, (2017) 60:16:6998 | ||||
Kd | 6.39 | MedChemComm, (2016) 7:12:2246 | ||||
IC50 | 6 | J Med Chem, (2017) 60:16:6998 | ||||
IC50 | 6 | Journal of Medicinal Chemistry, (2017) None:16:6998 | ||||
BRD1
Bromodomain-containing protein 1
8 Activities
Items per page:
1 – 8 of 8
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 6.97 | |||||
IC50 | 7.34 | J Med Chem, (2017) 60:16:6998 | ||||
Kd | 6.97 | MedChemComm, (2015) 6:9:1587 | ||||
Kd | 6.97 | MedChemComm, (2016) 7:12:2246 | ||||
Kd | 6.96 | J. Med. Chem., (2016) 59:4:1271 | ||||
Kd | 6.96 | J Med Chem, (2017) 60:16:6998 | ||||
IC50 | 6.5 | Journal of Medicinal Chemistry, (2017) None:16:6998 | ||||
IC50 | 6.21 | J Med Chem, (2017) 60:16:6998 | ||||
BRD9
Bromodomain-containing protein 9
2 Activities
BRD7
Bromodomain-containing protein 7
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.85 | J Med Chem, (2017) 60:16:6998 | ||||