Pharos : Ligand Details - 41TSVPX15U1P

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: TAK-901

PubChem: 16124208

ChEMBL: CHEMBL3544932

LyCHI: 41TSVPX15U1P

Target Activities

Explore Associated and Predicted Targets

AURKA

Tchem

Aurora kinase A

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	7.85		None, None:None:None

Kd	7.62		Science, (2017) 358:6367:None	29191878

PRKAG2

Tchem

5'-AMP-activated protein kinase subunit gamma-2

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	6.29		Science, (2017) 358:6367:None	29191878

YES1

Tclin

Tyrosine-protein kinase Yes

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	7.66		Science, (2017) 358:6367:None	29191878

EPHA4

Tchem

Ephrin type-A receptor 4

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	7.66		Science, (2017) 358:6367:None	29191878

IRAK3

Tchem

Interleukin-1 receptor-associated kinase 3

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	7.57		Science, (2017) 358:6367:None	29191878

BCR

Tclin

Breakpoint cluster region protein

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	6.88		Science, (2017) 358:6367:None	29191878

ERCC2

Tchem

General transcription and DNA repair factor IIH helicase subunit XPD

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	6.61		Science, (2017) 358:6367:None	29191878