TAK-901
Ligand Summary
Target Activities
AURKA
Aurora kinase A
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.85 | None, None:None:None | ||||
Kd | 7.62 | Science, (2017) 358:6367:None | ||||
PRKAG2
5'-AMP-activated protein kinase subunit gamma-2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 6.29 | Science, (2017) 358:6367:None | ||||
YES1
Tyrosine-protein kinase Yes
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.66 | Science, (2017) 358:6367:None | ||||
EPHA4
Ephrin type-A receptor 4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.66 | Science, (2017) 358:6367:None | ||||
IRAK3
Interleukin-1 receptor-associated kinase 3
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.57 | Science, (2017) 358:6367:None | ||||
BCR
Breakpoint cluster region protein
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 6.88 | Science, (2017) 358:6367:None | ||||
ERCC2
General transcription and DNA repair factor IIH helicase subunit XPD
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 6.61 | Science, (2017) 358:6367:None | ||||