SAR260301
Ligand Summary
Name: SAR260301
PubChem: 49854424
PubChem: 135565159
Guide to Pharmacology: 8793
ChEMBL: CHEMBL3112866
LyCHI: 3W776L4SJ9VG
Target Activities
AKT1
RAC-alpha serine/threonine-protein kinase
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.3 | None, (2015) None:None:None | ||||
IC50 | 8.05 | None, (2015) None:None:None | ||||
IC50 | 7.8 | None, (2015) None:None:None | ||||
IC50 | 7.72 | None, (2015) None:None:None | ||||
IC50 | 7.57 | None, (2015) None:None:None | ||||
PIK3CB
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
2 Activities
PIK3C3
Phosphatidylinositol 3-kinase catalytic subunit type 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.74 | |||||
PIK3CA
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 5.81 | |||||
PIK3CD
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.33 | |||||
PIK3C2G
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 5.42 | |||||