CHEMBL2153434
Ligand Summary
Name: benzyl 1-methyl-6-phenyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-ylcarbamate
PubChem: 13953710
Guide to Pharmacology: 7514
ChEMBL: CHEMBL2153434
LyCHI: 3RVZJBMCTHN6
Target Activities
Items per page:
10
1 – 3 of 3
BRD2
Bromodomain-containing protein 2
8 Activities
Items per page:
1 – 8 of 8
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 6.66 | J. Med. Chem., (2011) 54:11:3827 | ||||
Kd | 7.27 | J. Med. Chem., (2011) 54:11:3827 | ||||
Kd | 7.28 | J. Med. Chem., (2011) 54:11:3827 | ||||
Kd | 7.28 | J. Med. Chem., (2011) 54:11:3827 | ||||
Kd | 7.34 | J. Med. Chem., (2011) 54:11:3827 | ||||
IC50 | 7.52 | J. Med. Chem., (2011) 54:11:3827 | ||||
Kd | 7.72 | J. Med. Chem., (2011) 54:11:3827 | ||||
IC50 | 7.51999998 | |||||