US9255106, S3
Ligand Summary
Target Activities
PARP1
Poly [ADP-ribose] polymerase 1
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9.13 | None, (2016) None:None:None | ||||
IC50 | 9.13 | Eur J Med Chem, (2019) 165:None:198 | ||||
IC50 | 8.76 | Eur J Med Chem, (2019) 165:None:198 | ||||
IC50 | 8 | None, (2016) None:None:None | ||||
IC50 | 7.76 | None, (2016) None:None:None | ||||
PARP2
Poly [ADP-ribose] polymerase 2
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9.66 | None, (2016) None:None:None | ||||
IC50 | 9.66 | Eur J Med Chem, (2019) 165:None:198 | ||||
TNKS
Tankyrase-1
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.43 | None, (2016) None:None:None | ||||
IC50 | 6.19 | None, (2016) None:None:None | ||||
PARP3
Poly [ADP-ribose] polymerase 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.17 | None, (2016) None:None:None | ||||
TNKS2
Tankyrase-2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.03 | None, (2016) None:None:None | ||||