Pharos : Ligand Details - 3MT2D61G16Y1

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: US9255106, S3

PubChem: 72736758

ChEMBL: CHEMBL3907010

LyCHI: 3MT2D61G16Y1

Target Activities

PARP1

Tclin

Poly [ADP-ribose] polymerase 1

5 Activities

Items per page:

1 – 5 of 5

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	9.13		None, (2016) None:None:None

IC50	9.13		Eur J Med Chem, (2019) 165:None:198	30684797

IC50	8.76		Eur J Med Chem, (2019) 165:None:198	30684797

IC50	8		None, (2016) None:None:None

IC50	7.76		None, (2016) None:None:None

PARP2

Tclin

Poly [ADP-ribose] polymerase 2

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	9.66		None, (2016) None:None:None

IC50	9.66		Eur J Med Chem, (2019) 165:None:198	30684797

TNKS

Tchem

Tankyrase-1

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.43		None, (2016) None:None:None

IC50	6.19		None, (2016) None:None:None

PARP3

Tclin

Poly [ADP-ribose] polymerase 3

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.17		None, (2016) None:None:None

TNKS2

Tchem

Tankyrase-2

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.03		None, (2016) None:None:None