CHEMBL233421
Ligand Summary
Name: 4-(2-aza-bicyclo[2.2.1]heptan-2-ylmethyl)-N-(2-methoxyphenethyl)-N-(pyrrolidin-3-yl)benzamide
PubChem: 44433050
ChEMBL: CHEMBL233421
LyCHI: 3BKVQCTM9U4Q
Target Activities
MBTPS1
Membrane-bound transcription factor site-1 protease
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.02 | Bioorg. Med. Chem. Lett., (2007) 17:16:4411 | ||||