Pharos : Ligand Details - 2S966G8W6KCU

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: Cdk1/2 inhibitor III

PubChem: 5330812

Guide to Pharmacology: 5946

ChEMBL: CHEMBL261720

LyCHI: 2S966G8W6KCU

Target Activities

Explore Associated and Predicted Targets

CDK1

Tchem

Cyclin-dependent kinase 1

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	9.22			15974571

CDK2

Tchem

Cyclin-dependent kinase 2

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	9.3			15974571

FLT1

Tclin

Vascular endothelial growth factor receptor 1

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.49			15974571

CLK1

Tchem

Dual specificity protein kinase CLK1

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	8.05		Eur J Med Chem, (2017) 126:None:754	27940419

CLK3

Tchem

Dual specificity protein kinase CLK3

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.54		Eur J Med Chem, (2017) 126:None:754	27940419