CHEMBL249097
Ligand Summary
Name: 3-(4-(5-hydroxy-2-methylphenylamino)pyrimidin-2-ylamino)benzamide
PubChem: 25138012
ChEMBL: CHEMBL249097
LyCHI: 2NH7CFPSTX42
Target Activities
TXK
Tyrosine-protein kinase TXK
2 Activities
BLK
Tyrosine-protein kinase Blk
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 9 | J. Med. Chem., (2008) 51:24:7898 | ||||
FYN
Tyrosine-protein kinase Fyn
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 9.4 | J. Med. Chem., (2008) 51:24:7898 | ||||
LCK
Tyrosine-protein kinase Lck
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.85 | Bioorg. Med. Chem. Lett., (2007) 17:15:4363 | ||||
EPHA2
Ephrin type-A receptor 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.1 | J. Med. Chem., (2008) 51:24:7898 | ||||
YES1
Tyrosine-protein kinase Yes
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 9 | J. Med. Chem., (2008) 51:24:7898 | ||||
SYK
Tyrosine-protein kinase SYK
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.58 | Bioorg. Med. Chem. Lett., (2007) 17:15:4363 | ||||
CSK
Tyrosine-protein kinase CSK
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.55 | J. Med. Chem., (2008) 51:24:7898 | ||||
LYN
Tyrosine-protein kinase Lyn
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.52 | Bioorg. Med. Chem. Lett., (2007) 17:15:4363 | ||||
EPHB2
Ephrin type-B receptor 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.15 | J. Med. Chem., (2008) 51:24:7898 | ||||
EPHA5
Ephrin type-A receptor 5
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.52 | J. Med. Chem., (2008) 51:24:7898 | ||||
EPHA4
Ephrin type-A receptor 4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.3 | J. Med. Chem., (2008) 51:24:7898 | ||||
FGR
Tyrosine-protein kinase Fgr
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 9.52 | J. Med. Chem., (2008) 51:24:7898 | ||||
EPHA6
Ephrin type-A receptor 6
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.7 | J. Med. Chem., (2008) 51:24:7898 | ||||
PTK6
Protein-tyrosine kinase 6
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.7 | J. Med. Chem., (2008) 51:24:7898 | ||||
EPHA3
Ephrin type-A receptor 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 10 | J. Med. Chem., (2008) 51:24:7898 | ||||
BTK
Tyrosine-protein kinase BTK
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.05 | Bioorg. Med. Chem. Lett., (2007) 17:15:4363 | ||||
EPHA1
Ephrin type-A receptor 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.3 | J. Med. Chem., (2008) 51:24:7898 | ||||