Pharos: Illuminating the Druggable Genome

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Ligand Summary

Ligand Structure

chemical structure image

Synonyms & Links

NCATS Inxight: Drugs: 96607511

Name: 2-(2-Aminothiazol-4-yl)isonicotinic Acid

PubChem: 96607511

ChEMBL: CHEMBL3774692

LyCHI: 2C5PS77SCTBP

Target Activities

Items per page:

10

1 – 6 of 6

KDM4A

Tchem

Lysine-specific demethylase 4A

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.7		J. Med. Chem., (2016) 59:4:1388	26741168

KDM4B

Tchem

Lysine-specific demethylase 4B

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.08		J. Med. Chem., (2016) 59:4:1388	26741168

KDM3A

Tchem

Lysine-specific demethylase 3A

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.24		J. Med. Chem., (2016) 59:4:1388	26741168

KDM5C

Tchem

Lysine-specific demethylase 5C

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.92		J. Med. Chem., (2016) 59:4:1388	26741168

KDM5B

Tchem

Lysine-specific demethylase 5B

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.92		J. Med. Chem., (2016) 59:4:1388	26741168

KDM6B

Tchem

Lysine-specific demethylase 6B

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6		J. Med. Chem., (2016) 59:4:1388	26741168