CHEMBL3220922
Ligand Summary
Name: Isopropyl((2S,4R)-1-acetyl-6-(4-(8-(hydroxyamino)-8-oxooctanamido)phenyl)-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)carbamate
PubChem: 90667452
ChEMBL: CHEMBL3220922
LyCHI: 282VQZPBN1JV
Target Activities
BRD4
Bromodomain-containing protein 4
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.3 | MedChemComm, (2014) 5:3:342 | ||||
Kd | 7.28 | MedChemComm, (2014) 5:3:342 | ||||
Kd | 7.24 | MedChemComm, (2014) 5:3:342 | ||||
Kd | 6.95 | MedChemComm, (2014) 5:3:342 | ||||
HDAC1
Histone deacetylase 1
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.6 | MedChemComm, (2014) 5:3:342 | ||||
Kd | 6.48 | MedChemComm, (2014) 5:3:342 | ||||
HDAC6
Histone deacetylase 6
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 6.63 | MedChemComm, (2014) 5:3:342 | ||||
IC50 | 6.38 | MedChemComm, (2014) 5:3:342 | ||||
HDAC3
Histone deacetylase 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 6.37 | MedChemComm, (2014) 5:3:342 | ||||
HDAC8
Histone deacetylase 8
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 6.48 | MedChemComm, (2014) 5:3:342 | ||||
HDAC10
Histone deacetylase 10
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 6.68 | MedChemComm, (2014) 5:3:342 | ||||
BRD2
Bromodomain-containing protein 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.5 | MedChemComm, (2014) 5:3:342 | ||||
BRD3
Bromodomain-containing protein 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.16 | MedChemComm, (2014) 5:3:342 | ||||
HDAC2
Histone deacetylase 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 6.02 | MedChemComm, (2014) 5:3:342 | ||||