CHEMBL495727
Ligand Summary
Name: 1-Cyclopropyl-3-[3-(5-morpholin-4-ylmethyl-1H-benzoimidazol-2-yl)-1H-pyrazol-4-yl]urea
PubChem: 135398495
ChEMBL: CHEMBL495727
LyCHI: 25G2CWCX84YS
Target Activities
Items per page:
10
1 – 10 of 23
JAK3
Tyrosine-protein kinase JAK3
2 Activities
JAK2
Tyrosine-protein kinase JAK2
2 Activities
AURKA
Aurora kinase A
2 Activities
AURKB
Aurora kinase B
2 Activities
FLT3
Receptor-type tyrosine-protein kinase FLT3
2 Activities
RPS6KA3
Ribosomal protein S6 kinase alpha-3
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 9 | J. Med. Chem., (2009) 52:2:379 | ||||
RPS6KA2
Ribosomal protein S6 kinase alpha-2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 9 | J. Med. Chem., (2009) 52:2:379 | ||||
GSK3B
Glycogen synthase kinase-3 beta
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 9 | J. Med. Chem., (2009) 52:2:379 | ||||
FGFR2
Fibroblast growth factor receptor 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 9 | J. Med. Chem., (2009) 52:2:379 | ||||
YES1
Tyrosine-protein kinase Yes
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 9 | J. Med. Chem., (2009) 52:2:379 | ||||