AT-9283
Ligand Summary
Target Activities
ABL1
Tyrosine-protein kinase ABL1
3 Activities
JAK2
Tyrosine-protein kinase JAK2
3 Activities
FGFR1
Fibroblast growth factor receptor 1
3 Activities
AURKB
Aurora kinase B
3 Activities
AURKA
Aurora kinase A
3 Activities
FLT3
Receptor-type tyrosine-protein kinase FLT3
2 Activities
JAK3
Tyrosine-protein kinase JAK3
2 Activities
FGFR2
Fibroblast growth factor receptor 2
2 Activities
GSK3B
Glycogen synthase kinase-3 beta
2 Activities
RET
Proto-oncogene tyrosine-protein kinase receptor Ret
2 Activities
RPS6KA3
Ribosomal protein S6 kinase alpha-3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9 | J. Med. Chem., (2009) 52:2:379 | ||||
PRKAG2
5'-AMP-activated protein kinase subunit gamma-2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.21 | Science, (2017) 358:6367:None | ||||
FLT1
Vascular endothelial growth factor receptor 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8 | J. Med. Chem., (2009) 52:2:379 | ||||
FLT4
Vascular endothelial growth factor receptor 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9 | J. Med. Chem., (2009) 52:2:379 | ||||
PDGFRA
Platelet-derived growth factor receptor alpha
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8 | J. Med. Chem., (2009) 52:2:379 | ||||
SRC
Proto-oncogene tyrosine-protein kinase Src
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8 | J. Med. Chem., (2009) 52:2:379 | ||||
KDR
Vascular endothelial growth factor receptor 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8 | J. Med. Chem., (2009) 52:2:379 | ||||
YES1
Tyrosine-protein kinase Yes
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9 | J. Med. Chem., (2009) 52:2:379 | ||||
RPS6KA4
Ribosomal protein S6 kinase alpha-4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8 | J. Med. Chem., (2009) 52:2:379 | ||||
FGFR3
Fibroblast growth factor receptor 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8 | J. Med. Chem., (2009) 52:2:379 | ||||
GSK3A
Glycogen synthase kinase-3 alpha
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.22 | Science, (2017) 358:6367:None | ||||
AAK1
AP2-associated protein kinase 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.77 | Science, (2017) 358:6367:None | ||||
PRKD1
Serine/threonine-protein kinase D1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8 | J. Med. Chem., (2009) 52:2:379 | ||||
RPS6KA2
Ribosomal protein S6 kinase alpha-2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9 | J. Med. Chem., (2009) 52:2:379 | ||||
TYK2
Non-receptor tyrosine-protein kinase TYK2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9 | J. Med. Chem., (2009) 52:2:379 | ||||
MET
Hepatocyte growth factor receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.15 | Science, (2017) 358:6367:None | ||||
STK17A
Serine/threonine-protein kinase 17A
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8 | J. Med. Chem., (2009) 52:2:379 | ||||
EPHA7
Ephrin type-A receptor 7
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.1 | Science, (2017) 358:6367:None | ||||
PDK1
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8 | J. Med. Chem., (2009) 52:2:379 | ||||
RPS6KA6
Ribosomal protein S6 kinase alpha-6
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.8 | Science, (2017) 358:6367:None | ||||
BCR
Breakpoint cluster region protein
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 6.81 | Science, (2017) 358:6367:None | ||||
ACVRL1
Serine/threonine-protein kinase receptor R3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.82 | Science, (2017) 358:6367:None | ||||
MERTK
Tyrosine-protein kinase Mer
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9 | J. Med. Chem., (2009) 52:2:379 | ||||
BMPR1B
Bone morphogenetic protein receptor type-1B
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.68 | Science, (2017) 358:6367:None | ||||
PRKACG
cAMP-dependent protein kinase catalytic subunit gamma
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.52 | Science, (2017) 358:6367:None | ||||
CDK10
Cyclin-dependent kinase 10
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.05 | Science, (2017) 358:6367:None | ||||
ACAD10
Acyl-CoA dehydrogenase family member 10
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 6.84 | Science, (2017) 358:6367:None | ||||
Q6ZSR9
Uncharacterized protein FLJ45252
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.62 | Science, (2017) 358:6367:None | ||||
PLK4
Serine/threonine-protein kinase PLK4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.68 | Science, (2017) 358:6367:None | ||||
EPHB6
Ephrin type-B receptor 6
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.92 | Science, (2017) 358:6367:None | ||||