CHEMBL214239
Ligand Summary
Name: N-(3,5-diamino-6-chloropyrazine-2-carbonyl)-N'-[4-(4-hydroxymethylphenyl)-butyl]guanidine
PubChem: 10237531
ChEMBL: CHEMBL214239
LyCHI: 1ZJQX9VYT6UG
Target Activities
SCNN1A
Amiloride-sensitive sodium channel subunit alpha
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.85 | J. Med. Chem., (2006) 49:14:4098 | ||||