XL-228
Ligand Summary
Target Activities
FYN
Tyrosine-protein kinase Fyn
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.64 | Science, (2017) 358:6367:None | ||||
FLT3
Receptor-type tyrosine-protein kinase FLT3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.3 | Science, (2017) 358:6367:None | ||||
PTK2
Focal adhesion kinase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Kd | 7.66 | Science, (2017) 358:6367:None | ||||
NTRK1
High affinity nerve growth factor receptor
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Kd | 8.22 | Science, (2017) 358:6367:None | ||||
FGFR1
Fibroblast growth factor receptor 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.05 | Science, (2017) 358:6367:None | ||||
ABL2
Tyrosine-protein kinase ABL2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.1 | Science, (2017) 358:6367:None | ||||
BMP2K
BMP-2-inducible protein kinase
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.85 | Science, (2017) 358:6367:None | ||||
EPHA7
Ephrin type-A receptor 7
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.77 | Science, (2017) 358:6367:None | ||||
BCR
Breakpoint cluster region protein
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.52 | Science, (2017) 358:6367:None | ||||
TNK1
Non-receptor tyrosine-protein kinase TNK1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.52 | Science, (2017) 358:6367:None | ||||
CDK17
Cyclin-dependent kinase 17
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.3 | Science, (2017) 358:6367:None | ||||
MAP4K1
Mitogen-activated protein kinase kinase kinase kinase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.82 | Science, (2017) 358:6367:None | ||||
ACVR1
Activin receptor type-1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.3 | Science, (2017) 358:6367:None | ||||
AURKB
Aurora kinase B
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.4 | Science, (2017) 358:6367:None | ||||
ERCC2
General transcription and DNA repair factor IIH helicase subunit XPD
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 6.02 | Science, (2017) 358:6367:None | ||||
AURKA
Aurora kinase A
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.52 | Science, (2017) 358:6367:None | ||||
Uncharacterized protein FLJ45252
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Kd | 6.69 | Science, (2017) 358:6367:None | ||||
EPHA1
Ephrin type-A receptor 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.3 | Science, (2017) 358:6367:None | ||||
RET
Proto-oncogene tyrosine-protein kinase receptor Ret
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.05 | Science, (2017) 358:6367:None | ||||
PLK4
Serine/threonine-protein kinase PLK4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.52 | Science, (2017) 358:6367:None | ||||
PKN1
Serine/threonine-protein kinase N1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.96 | Science, (2017) 358:6367:None | ||||
EPHB6
Ephrin type-B receptor 6
1 Activities
Items per page:
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.58 | Science, (2017) 358:6367:None | ||||