SID103905191
Ligand Summary
Target Activities
MAPK8
Mitogen-activated protein kinase 8
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.4 | None, None:None:None | ||||
IC50 | 8.33 | ACS Med. Chem. Lett., (2012) 3:7:560 | ||||
IC50 | 7.72 | J. Med. Chem., (2006) 49:15:4455 | ||||
IC50 | 7.72 | Bioorg. Med. Chem. Lett., (2007) 17:2:495 | ||||
MAPK10
Mitogen-activated protein kinase 10
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.6 | None, None:None:None | ||||
MAPK9
Mitogen-activated protein kinase 9
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.9 | None, None:None:None | ||||
JUN
Transcription factor AP-1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
EC50 | 6.5 | Bioorg. Med. Chem. Lett., (2007) 17:2:495 | ||||
RPS27
40S ribosomal protein S27
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.25 | ACS Med. Chem. Lett., (2012) 3:7:560 | ||||