Pharos : Ligand Details - 1AGP8HVPT6UW

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: 2-Chloro-4-(5-(2,6-difluoro-3-hydroxybenzoyl)thiophen-2-yl)phenyl sulfamate

PubChem: 137638205

ChEMBL: CHEMBL4071245

LyCHI: 1AGP8HVPT6UW

Target Activities

Explore Associated and Predicted Targets

STS

Tchem

Steryl-sulfatase

3 Activities

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1 – 3 of 3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.81		J Med Chem, (2017) 60:9:4086	28406629

IC50	7.79		J Med Chem, (2017) 60:9:4086	28406629

IC50	6.84		J Med Chem, (2017) 60:9:4086	28406629

HSD17B1

Tchem

Estradiol 17-beta-dehydrogenase 1

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	8.96		J Med Chem, (2017) 60:9:4086	28406629

IC50	7.65		J Med Chem, (2017) 60:9:4086	28406629

HSD17B2

Tchem

Estradiol 17-beta-dehydrogenase 2

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.44		J Med Chem, (2017) 60:9:4086	28406629