tolvaptan
Ligand Summary
A benzazepine derivative and selective VASOPRESSIN V2 RECEPTOR antagonist that is used to treat euvolemic and hypervolemic HYPONATREMIA. It is also used in the treatment of rapidly progressing AUTOSOMAL DOMINANT POLYCYSTIC KIDNEY DISEASE to slow the rate of cyst development and renal insufficiency.
UNII: 21G72T1950
PubChem: 216237
Guide to Pharmacology: 2226
ChEMBL: CHEMBL344159
DrugCentral: 4110
LyCHI: JCWBL5XZ9URG
Target Activities
7 Activities
Items per page:
1 – 7 of 7
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