timolol
Ligand Summary
A beta-adrenergic antagonist that is similar in action to PROPRANOLOL; the levo-isomer is more active. Timolol has been proposed as an anti-hypertensive, anti-arrhythmic, anti-angina, and anti-glaucoma agent. It is also used in the treatment of MIGRAINE DISORDERS and tremor.
UNII: 5JKY92S7BR
PubChem: 33624
Guide to Pharmacology: 565
ChEMBL: CHEMBL499
DrugCentral: 4061
LyCHI: 952J8AXNZB3W
Target Activities
9 Activities
Items per page:
1 – 9 of 9
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
- | ||||||
Ki | ||||||
IC50 | ||||||
Ki | ||||||
Ki | ||||||
Ki | ||||||
IC50 | ||||||
Ki | ANTAGONIST | |||||
Ki | ANTAGONIST | |||||