tapentadol
Ligand Summary
An opioid analgesic, MU OPIOID RECEPTOR agonist, and noradrenaline reuptake inhibitor that is used in the treatment of moderate to severe pain, and of pain associated with DIABETIC NEUROPATHIES.
UNII: H8A007M585
PubChem: 9838022
Guide to Pharmacology: 7477
ChEMBL: CHEMBL1201776
DrugCentral: 4283
LyCHI: LFH5DAQJQJMG
Target Activities
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | ||||||
Ki | ||||||
Ki | AGONIST | |||||
Ki | INHIBITOR | |||||