methysergide
Ligand Summary
An ergot derivative that is a congener of LYSERGIC ACID DIETHYLAMIDE. It antagonizes the effects of serotonin in blood vessels and gastrointestinal smooth muscle, but has few of the properties of other ergot alkaloids. Methysergide is used prophylactically in migraine and other vascular headaches and to antagonize serotonin in the carcinoid syndrome.
UNII: XZA9HY6Z98
PubChem: 9681
PubChem: 5281073
Guide to Pharmacology: 134
ChEMBL: CHEMBL1065
ChEMBL: CHEMBL1200938
DrugCentral: 1775
LyCHI: 3M5UQBRT98CD
Target Activities
29 Activities
Items per page:
1 – 10 of 29
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