macitentan
Ligand Summary
an endothelin receptor antagonist that prevents the binding of ET-1 to both ETA and ETB receptors, macitentan displays high affinity and sustained occupancy of the ET receptors in human pulmonary arterial smooth muscle cells
UNII: Z9K9Y9WMVL
PubChem: 16004692
Guide to Pharmacology: 7352
ChEMBL: CHEMBL2103873
DrugCentral: 4809
LyCHI: RCSNMFR4CQSF
Target Activities
7 Activities
Items per page:
1 – 7 of 7
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