isradipine
Ligand Summary
A potent antagonist of CALCIUM CHANNELS that is highly selective for VASCULAR SMOOTH MUSCLE. It is effective in the treatment of chronic stable angina pectoris, hypertension, and congestive cardiac failure.
UNII: YO1UK1S598
PubChem: 13773524
PubChem: 3784
Guide to Pharmacology: 4488
ChEMBL: CHEMBL399539
ChEMBL: CHEMBL1648
DrugCentral: 1511
LyCHI: ZC55D4516PJZ
Target Activities
8 Activities
Items per page:
1 – 8 of 8
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
- | ||||||
- | ||||||
- | ||||||
IC50 | ||||||
- | ||||||
IC50 | ||||||
IC50 | GATING INHIBITOR | |||||
IC50 | GATING INHIBITOR | |||||