gabapentin enacarbil
Ligand Summary
Gabapentin enacarbil is a prodrug of gabapentin and, accordingly, its therapeutic effects in restless legs syndrome and postherpetic neuralgia are attributable to gabapentin. In animal models of analgesia, gabapentin prevents allodynia (pain-related behavior in response to a normally innocuous stimulus) and hyperalgesia (exaggerated response to painful stimuli).
UNII: 75OCL1SPBQ
PubChem: 9883933
ChEMBL: CHEMBL1628502
DrugCentral: 4177
LyCHI: 81W8SQNQMY9A
Target Activities
2 Activities
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