flibanserin
Ligand Summary
a serotonin receptor modulator with high affinity for the following serotonin (5-hydroxytryptamine or 5-T) receptors: agonist activity at 5-HT1A and antagonist activity at 5-HT2A. Flibanserin also has moderate antagonist activities at the 5-HT2B, 5-HT2C, and dopamine D4 receptors, used in the treatment of premenopausal women with hypoactive sexual desire disorder
UNII: 37JK4STR6Z
PubChem: 6918248
Guide to Pharmacology: 8182
ChEMBL: CHEMBL231068
DrugCentral: 5022
LyCHI: GR23QZKJ5F95
Target Activities
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | ||||||
Ki | ||||||
Ki | AGONIST | |||||
Ki | ANTAGONIST | |||||
Ki | ANTAGONIST | |||||