droperidol
Ligand Summary
A butyrophenone with general properties similar to those of HALOPERIDOL. It is used in conjunction with an opioid analgesic such as FENTANYL to maintain the patient in a calm state of neuroleptanalgesia with indifference to surroundings but still able to cooperate with the surgeon. It is also used as a premedicant, as an antiemetic, and for the control of agitation in acute psychoses. (From Martindale, The Extra Pharmacopoeia, 29th ed, p593)
UNII: O9U0F09D5X
PubChem: 3168
ChEMBL: CHEMBL1108
DrugCentral: 966
LyCHI: SKWTUHL8J97Y
Target Activities
21 Activities
Items per page:
1 – 10 of 21
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | ||||||
IC50 | ||||||
Ki | ||||||
IC50 | ||||||
Ki | ||||||
IC50 | ||||||
Ki | ||||||
IC50 | ||||||
IC50 | ||||||
IC50 | ||||||