crisaborole
Ligand Summary
Crisaborole is a phosphodiesterase 4 (PDE-4) inhibitor. PDE-4 inhibition results in increased intracellular cyclic adenosine monophosphate (cAMP) levels. The specific mechanism(s) by which crisaborole exerts its therapeutic action for the treatment of atopic dermatitis is not well defined.
UNII: Q2R47HGR7P
PubChem: 44591583
Guide to Pharmacology: 9151
ChEMBL: CHEMBL484785
DrugCentral: 5201
LyCHI: WY8BUK2X33RS
Target Activities
13 Activities
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