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azelastine

Ligand Summary
Ligand Structure
Rendered image for the query structure
Description
Azelastine hydrochloride, a phthalazinone derivative, exhibits histamine H1-receptor antagonist activity in isolated tissues, animal models, and humans. Azelastine Hydrochloride is administered as a racemic mixture with no difference in pharmacologic activity noted between the enantiomers in in vitro studies. The major metabolite, desmethylazelastine, also possesses H1-receptor antagonist activity.
Synonyms & Links
PubChem: 2267
Guide to Pharmacology: 7121
DrugCentral: 271
LyCHI:  VKY49BVV56A6


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Target Activities