imatinib
Ligand Summary
A tyrosine kinase inhibitor and ANTINEOPLASTIC AGENT that inhibits the BCR-ABL kinase created by chromosome rearrangements in CHRONIC MYELOID LEUKEMIA and ACUTE LYMPHOBLASTIC LEUKEMIA, as well as PDG-derived tyrosine kinases that are overexpressed in gastrointestinal stromal tumors.
UNII: BKJ8M8G5HI
PubChem: 5291
Guide to Pharmacology: 5687
ChEMBL: CHEMBL941
DrugCentral: 1423
LyCHI: VLU17BQBSGWU
Target Activities
86 Activities
Items per page:
1 – 10 of 86
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