carvedilol
Ligand Summary
A carbazole and propanol derivative that acts as a non-cardioselective beta blocker and vasodilator. It has blocking activity for ALPHA 1 ADRENERGIC RECEPTORS and, at higher doses, may function as a blocker of CALCIUM CHANNELS; it also has antioxidant properties. Carvedilol is used in the treatment of HYPERTENSION; ANGINA PECTORIS; and HEART FAILURE. It can also reduce the risk of death following MYOCARDIAL INFARCTION.
UNII: 0K47UL67F2
PubChem: 2585
Guide to Pharmacology: 551
ChEMBL: CHEMBL723
DrugCentral: 522
LyCHI: BM9MKM694U27
Target Activities
33 Activities
Items per page:
1 – 10 of 33
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